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Compound Detail

CHEMBL423111

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CCc1ccccc1C1Cc2cc(OC(=O)C3O[C@@H](O)[C@H](O)[C@@H](O)[C@H]3O)c(CCCOc3ccccc3)cc2O1

Basic Information

ChEMBL ID CHEMBL423111
Phase Preclinical
Structure Type MOL
InChI Key OAQOWYUAUPSECR-GAAWIUQDSA-N
0
Targets
0
Activities
0
Assay Types
1
PK Parameters
3
Publications
0
Known Names

Molecular Properties

550.6
MW (Da)
2.64
ALogP
9
HBA
4
HBD
134.9
PSA (Ų)
0.18
QED
1
Ro5 Violations
9
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C31H34O9
MW 550.60
Aromatic Rings 3
Heavy Atoms 40
NP-Likeness 0.65

Pharmacokinetic Data

Parameter Value Units Species
F - % -

Literature References

PubMed DOI Target Context # Activities
1313879 10.1021/jm00085a019 Rattus norvegicus 4
1313879 10.1021/jm00085a019 Leukotriene B4 receptor 1 1
1313879 10.1021/jm00085a019 ADMET 1

Data from ChEMBL 36 via Core Engine