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Compound Detail

CHEMBL430496

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CCNC(=O)C[C@H](NC(=O)[C@@H](NC(=O)C(CC)CC)C(C)(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)O

Basic Information

ChEMBL ID CHEMBL430496
Phase Preclinical
Structure Type MOL
InChI Key NIFNUTIJWSPFNB-ZVVDCOBXSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

599.7
MW (Da)
0.54
ALogP
7
HBA
7
HBD
220.1
PSA (Ų)
0.12
QED
2
Ro5 Violations
18
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H49N5O9
MW 599.73
Aromatic Rings 0
Heavy Atoms 42
NP-Likeness 0.21

Activity Summary

IC50 1 meas. best 5.16

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.16 5.16 6900.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 6900.0 nM 5.16 Inhibition of Herpes simplex virus type 1 ribonucleotide reductase 8411018

Literature References

PubMed DOI Target Context # Activities
8411018 10.1021/jm00072a021 Unchecked 1

Data from ChEMBL 36 via Core Engine