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Compound Detail

CHEMBL438499

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CCCCCCCCCCCCOC(=O)[C@@H](C)[C@@]1(O)[C@@H](O[C@@H]2OC[C@H](O)[C@H](OC/C=C\CCCCCCCCOC(=O)c3ccc(OC)cc3)[C@H]2OC(=O)c2ccc(OC)cc2)C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@@]21C

Basic Information

ChEMBL ID CHEMBL438499
Phase Preclinical
Structure Type MOL
InChI Key MLFJZHLSWWJFBK-WOYOLQPJSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

1115.5
MW (Da)

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C66H98O14
MW 1115.50

Literature References

PubMed DOI Target Context # Activities
17127060 10.1016/j.bmcl.2006.11.032 Jurkat 1
17127060 10.1016/j.bmcl.2006.11.032 RKO 1
17127060 10.1016/j.bmcl.2006.11.032 HeLa 1

Data from ChEMBL 36 via Core Engine