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Compound Detail

CHEMBL4453622

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O=C(C[C@H]1NCCC[C@@H]1O)Cn1cnc2c(c1=O)CCCC2

Basic Information

ChEMBL ID CHEMBL4453622
Phase Preclinical
Structure Type MOL
InChI Key ZMMDIKHKFCGQDK-CABCVRRESA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

305.4
MW (Da)
0.19
ALogP
6
HBA
2
HBD
84.2
PSA (Ų)
0.83
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H23N3O3
MW 305.38
Aromatic Rings 1
Heavy Atoms 22
NP-Likeness 0.31

Activity Summary

EC50 1 meas. best 6.06

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Toxoplasma gondii
CHEMBL612888
EC50 6.06 6.06 880.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Toxoplasma gondii EC50 = 880.0 nM 6.06 Antiparasitic activity against Toxoplasma gondii 31585276

Literature References

PubMed DOI Target Context # Activities
31585276 10.1016/j.ejmech.2019.111711 Toxoplasma gondii 1

Data from ChEMBL 36 via Core Engine