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Compound Detail

CHEMBL446672

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COCCOCn1c(N)c(C#N)c2c(N)ncnc21

Basic Information

ChEMBL ID CHEMBL446672
Phase Preclinical
Structure Type MOL
InChI Key CLQXQQWKOGUSCI-UHFFFAOYSA-N
1
Targets
3
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

262.3
MW (Da)
0.09
ALogP
8
HBA
2
HBD
125.0
PSA (Ų)
0.73
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C11H14N6O2
MW 262.27
Aromatic Rings 2
Heavy Atoms 19
NP-Likeness -1.23

Activity Summary

IC50 3 meas. best 5.09

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human betaherpesvirus 5
CHEMBL371
IC50 5.09 5.07 8200.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
8784444 10.1021/jm950835y Human betaherpesvirus 5 2
8784444 10.1021/jm950835y Human alphaherpesvirus 1 1
8784444 10.1021/jm950835y HFF 1
8784444 10.1021/jm950835y KB 1

Data from ChEMBL 36 via Core Engine