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Compound Detail

CHEMBL449731

NOROXYHYDRASTININE
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O=C1NCCc2cc3c(cc21)OCO3

Basic Information

ChEMBL ID CHEMBL449731
Name NOROXYHYDRASTININE
Phase Preclinical
Structure Type MOL
InChI Key VSOJKDUWYQCWFM-UHFFFAOYSA-N
0
Targets
1
Activities
1
Assay Types
0
PK Parameters
9
Publications
0
Known Names

Molecular Properties

191.2
MW (Da)
0.70
ALogP
3
HBA
1
HBD
47.6
PSA (Ų)
0.66
QED
0
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C10H9NO3
MW 191.19
Aromatic Rings 1
Heavy Atoms 14
NP-Likeness 0.87

Activity Summary

IC50 1 meas.

Literature References

PubMed DOI Target Context # Activities
- 10.1021/np50007a014 Staphylococcus aureus 1
- 10.1021/np50007a014 Escherichia coli 1
- 10.1021/np50007a014 Salmonella enterica subsp. enterica serovar Gallinarum 1
- 10.1021/np50007a014 Klebsiella pneumoniae 1
- 10.1021/np50007a014 Mycolicibacterium smegmatis 1
- 10.1021/np50007a014 Candida albicans 1
35286954 10.1016/j.bmc.2022.116705 MGC-803 1
35286954 10.1016/j.bmc.2022.116705 HGC-27 1
35286954 10.1016/j.bmc.2022.116705 GES1 1

Data from ChEMBL 36 via Core Engine