Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL4513472

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
CS(=O)(=O)[O-].O=C(Cc1ccc(O)c(O)c1)NCCCCCCCCCC[P+](c1ccccc1)(c1ccccc1)c1ccccc1

Basic Information

ChEMBL ID CHEMBL4513472
Phase Preclinical
Structure Type MOL
InChI Key BTOGKODBGNLZOT-UHFFFAOYSA-N
Parent Compound CHEMBL4596665
Active Moiety CHEMBL4596665
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

568.7
MW (Da)
6.87
ALogP
3
HBA
3
HBD
69.6
PSA (Ų)
0.08
QED
2
Ro5 Violations
16
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C37H46NO6PS
MW 663.82
Aromatic Rings 4
Heavy Atoms 41

Activity Summary

IC50 2 meas. best 4.55

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
No relevant target
CHEMBL2362975
IC50 4.55 4.4 28100.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
30784884 10.1016/j.ejmech.2019.01.055 SH-SY5Y 6
30784884 10.1016/j.ejmech.2019.01.055 No relevant target 5
30784884 10.1016/j.ejmech.2019.01.055 HepG2 3

Data from ChEMBL 36 via Core Engine