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Compound Detail

CHEMBL4516775

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CS(=O)(=O)[O-].O=C(Cc1cc(O)c(O)c(O)c1)NCCCCCCCCCC[P+](c1ccccc1)(c1ccccc1)c1ccccc1

Basic Information

ChEMBL ID CHEMBL4516775
Phase Preclinical
Structure Type MOL
InChI Key IXRZAJGKYZAWMH-UHFFFAOYSA-N
Parent Compound CHEMBL4598097
Active Moiety CHEMBL4598097
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

584.7
MW (Da)
6.58
ALogP
4
HBA
4
HBD
89.8
PSA (Ų)
0.07
QED
2
Ro5 Violations
16
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C37H46NO7PS
MW 679.82
Aromatic Rings 4
Heavy Atoms 42
NP-Likeness 0.05

Activity Summary

IC50 2 meas. best 5.12

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
No relevant target
CHEMBL2362975
IC50 5.12 4.9 7600.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
30784884 10.1016/j.ejmech.2019.01.055 SH-SY5Y 8
30784884 10.1016/j.ejmech.2019.01.055 No relevant target 5
30784884 10.1016/j.ejmech.2019.01.055 Unchecked 3
30784884 10.1016/j.ejmech.2019.01.055 HepG2 2

Data from ChEMBL 36 via Core Engine