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Compound Detail

CHEMBL4520942

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CC(=O)[C@@H]1CC[C@]2(C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CCC(=O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12

Basic Information

ChEMBL ID CHEMBL4520942
Phase Preclinical
Structure Type MOL
InChI Key KBNLDLGROQKYEQ-XFPNZXGSSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

426.7
MW (Da)
7.25
ALogP
2
HBA
0
HBD
34.1
PSA (Ų)
0.44
QED
1
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C29H46O2
MW 426.69
Aromatic Rings 0
Heavy Atoms 31
NP-Likeness 2.91

Activity Summary

IC50 1 meas. best 4.61

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Toxoplasma gondii
CHEMBL612888
IC50 4.61 4.61 24400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Toxoplasma gondii IC50 = 24400.0 nM 4.61 Antiparasitic activity against Toxoplasma gondii 31585276

Literature References

PubMed DOI Target Context # Activities
31585276 10.1016/j.ejmech.2019.111711 Toxoplasma gondii 1

Data from ChEMBL 36 via Core Engine