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Compound Detail

CHEMBL4546703

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CC(C)COc1cccc(Cl)c1-c1cc2cnc(N)nc2nc1N1C[C@@H]2[C@@H](N)[C@@H]2C1

Basic Information

ChEMBL ID CHEMBL4546703
Phase Preclinical
Structure Type MOL
InChI Key SLZBWLWZNBWUBK-QWHZDKJVSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
20
Publications
0
Known Names

Molecular Properties

424.9
MW (Da)
3.36
ALogP
7
HBA
2
HBD
103.2
PSA (Ų)
0.65
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H25ClN6O
MW 424.94
Aromatic Rings 3
Heavy Atoms 30
NP-Likeness -0.52

Literature References

PubMed DOI Target Context # Activities
31306011 10.1021/acs.jmedchem.9b00625 Pseudomonas aeruginosa 18
31306011 10.1021/acs.jmedchem.9b00625 Escherichia coli 7
31306011 10.1021/acs.jmedchem.9b00625 Epidermal growth factor receptor 1
31306011 10.1021/acs.jmedchem.9b00625 Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
31306011 10.1021/acs.jmedchem.9b00625 Casein kinase I isoform delta 1
31306011 10.1021/acs.jmedchem.9b00625 Cyclin-dependent kinase 1/cyclin B1 1
31306011 10.1021/acs.jmedchem.9b00625 Serine/threonine-protein kinase PAK 4 1
31306011 10.1021/acs.jmedchem.9b00625 Aurora kinase A 1
31306011 10.1021/acs.jmedchem.9b00625 Hepatocyte growth factor receptor 1
31306011 10.1021/acs.jmedchem.9b00625 Mitogen-activated protein kinase 14 1
31306011 10.1021/acs.jmedchem.9b00625 Mitogen-activated protein kinase 1 1
31306011 10.1021/acs.jmedchem.9b00625 High affinity nerve growth factor receptor 1
31306011 10.1021/acs.jmedchem.9b00625 Mitogen-activated protein kinase kinase kinase kinase 4 1
31306011 10.1021/acs.jmedchem.9b00625 Biotin carboxylase 1
31306011 10.1021/acs.jmedchem.9b00625 Fibroblast growth factor receptor 1 1
31306011 10.1021/acs.jmedchem.9b00625 Tyrosine-protein kinase BTK 1
31306011 10.1021/acs.jmedchem.9b00625 Proto-oncogene tyrosine-protein kinase Src 1
31306011 10.1021/acs.jmedchem.9b00625 Tyrosine-protein kinase Fyn 1
31306011 10.1021/acs.jmedchem.9b00625 Tyrosine-protein kinase ABL1 1
31306011 10.1021/acs.jmedchem.9b00625 Klebsiella pneumoniae 1

Data from ChEMBL 36 via Core Engine