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Compound Detail

CHEMBL455092

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COc1ccc(/C=C\c2cc(OC)c3c(c2)OCO3)cc1NC(=O)[C@H](C)[C@@H](OC)[C@@H]1CCCN1.O=C(O)C(F)(F)F

Basic Information

ChEMBL ID CHEMBL455092
Phase Preclinical
Structure Type MOL
InChI Key WQRWUUCMJDKGES-GASLPTIJSA-N
Parent Compound CHEMBL1186235
Active Moiety CHEMBL1186235
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
11
Publications
0
Known Names

Molecular Properties

468.6
MW (Da)
3.94
ALogP
7
HBA
2
HBD
87.3
PSA (Ų)
0.54
QED
0
Ro5 Violations
9
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H33F3N2O8
MW 582.57
Aromatic Rings 2
Heavy Atoms 34
NP-Likeness 0.71

Literature References

PubMed DOI Target Context # Activities
16124759 10.1021/np058033l SF-295 1
16124759 10.1021/np058033l NCI-H460 1
16124759 10.1021/np058033l MCF7 1
16124759 10.1021/np058033l KM-20L2 1
16124759 10.1021/np058033l BXPC-3 1
16124759 10.1021/np058033l DU-145 1
16124759 10.1021/np058033l Cryptococcus neoformans 1
16124759 10.1021/np058033l Neisseria gonorrhoeae 1
16124759 10.1021/np058033l Streptococcus pneumoniae 1
16124759 10.1021/np058033l Enterococcus faecalis 1
16124759 10.1021/np058033l P388 1

Data from ChEMBL 36 via Core Engine