Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL456220

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
CCCCCCCCCCCCCCCCCCOCCCOP(=O)([O-])CO[C@H](CO)Cn1ccc(N)nc1=O.[Na+]

Basic Information

ChEMBL ID CHEMBL456220
Phase Preclinical
Structure Type MOL
InChI Key FLSRPFRPLSTLMM-YCBFMBTMSA-M
Parent Compound CHEMBL1207921
Active Moiety CHEMBL1207921
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

589.8
MW (Da)
6.03
ALogP
9
HBA
3
HBD
146.1
PSA (Ų)
0.08
QED
2
Ro5 Violations
28
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C29H55N3NaO7P
MW 611.74
Aromatic Rings 1
Heavy Atoms 40
NP-Likeness 0.21

Activity Summary

IC50 1 meas. best 10.52

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human betaherpesvirus 5
CHEMBL371
IC50 10.52 10.52 0.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Human betaherpesvirus 5 IC50 = 0.03 nM 10.52 Antiviral activity against Human cytomegalovirus 19112024

Literature References

PubMed DOI Target Context # Activities
19112024 10.1016/j.bmc.2008.11.075 Human betaherpesvirus 5 1

Data from ChEMBL 36 via Core Engine