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Compound Detail

CHEMBL458737

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COC(=O)/C=C/[C@H](CC(C)C)NC(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)C(=O)NC(=O)[C@@H](N)C(C)C)C(N)=O

Basic Information

ChEMBL ID CHEMBL458737
Phase Preclinical
Structure Type MOL
InChI Key IAYNUBXUQUILHS-XQIKNGPFSA-N
0
Targets
0
Activities
0
Assay Types
1
PK Parameters
2
Publications
0
Known Names

Molecular Properties

652.8
MW (Da)
0.82
ALogP
9
HBA
6
HBD
228.9
PSA (Ų)
0.06
QED
2
Ro5 Violations
20
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C32H56N6O8
MW 652.83
Aromatic Rings 0
Heavy Atoms 46
NP-Likeness 0.35

Pharmacokinetic Data

Parameter Value Units Species
T1/2 1.957 hr Homo sapiens

Literature References

PubMed DOI Target Context # Activities
19250821 10.1016/j.bmcl.2009.02.046 Unchecked 3
19250821 10.1016/j.bmcl.2009.02.046 Plasma 1

Data from ChEMBL 36 via Core Engine