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Compound Detail

CHEMBL4647504

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CO[C@H]1[C@H](O[C@H]2CC[C@]3(C=O)[C@H]4CC[C@]5(C)[C@](O)(C6=CC(=O)OC6)CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)O[C@H](C)[C@H](O)[C@@H]1OC

Basic Information

ChEMBL ID CHEMBL4647504
Phase Preclinical
Structure Type MOL
InChI Key NERVBEHGMIDLEO-KFOBGKRGSA-N
0
Targets
1
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

594.7
MW (Da)
1.17
ALogP
11
HBA
4
HBD
161.2
PSA (Ų)
0.20
QED
2
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C31H46O11
MW 594.70
Aromatic Rings 0
Heavy Atoms 42
NP-Likeness 2.99

Activity Summary

IC50 1 meas.

Literature References

Data from ChEMBL 36 via Core Engine