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Compound Detail

CHEMBL4648754

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CO[C@H]1[C@H](O[C@H]2CC[C@]3(C=O)[C@H]4CC[C@]5(C)[C@@H]6CC[C@]5(O[C@H]5OC(=O)C[C@H]56)[C@@H]4CC[C@]3(O)C2)O[C@H](C)[C@H](O)[C@@H]1OC

Basic Information

ChEMBL ID CHEMBL4648754
Phase Preclinical
Structure Type MOL
InChI Key NLFMJFYKLJVIOT-DXQKBWEPSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

578.7
MW (Da)
2.50
ALogP
10
HBA
2
HBD
130.0
PSA (Ų)
0.29
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C31H46O10
MW 578.70
Aromatic Rings 0
Heavy Atoms 41
NP-Likeness 2.65

Literature References

PubMed DOI Target Context # Activities
31953129 10.1016/j.bmc.2019.115301 OVCAR-3 1
31953129 10.1016/j.bmc.2019.115301 Unchecked 1
31953129 10.1016/j.bmc.2019.115301 HT-29 1

Data from ChEMBL 36 via Core Engine