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Compound Detail

CHEMBL465159

PINUSOLIDIC ACID
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C=C1CC[C@@H]2[C@](C)(CCC[C@]2(C)C(=O)O)[C@H]1CCC1=CCOC1=O

Basic Information

ChEMBL ID CHEMBL465159
Name PINUSOLIDIC ACID
Phase Preclinical
Structure Type MOL
InChI Key FHQSDRHZGCMBKG-FIYPYCPBSA-N
1
Targets
2
Activities
2
Assay Types
0
PK Parameters
10
Publications
0
Known Names

Molecular Properties

332.4
MW (Da)
4.11
ALogP
3
HBA
1
HBD
63.6
PSA (Ų)
0.62
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C20H28O4
MW 332.44
Aromatic Rings 0
Heavy Atoms 24
NP-Likeness 3.48

Activity Summary

EC50 1 meas. best 5.33
IC50 1 meas.

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
SARS-CoV
CHEMBL4303836
EC50 5.33 5.33 4710.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
SARS-CoV EC50 = 4710.0 nM 5.33 Antiviral activity against SARS coronavirus in Vero E6 cells assessed as inhibit... 17663539

Literature References

PubMed DOI Target Context # Activities
17663539 10.1021/jm070295s SARS-CoV 5
15104493 10.1021/np034033e Erythrocyte 4
17663539 10.1021/jm070295s Vero 1
17663539 10.1021/jm070295s Unchecked 1
15104493 10.1021/np034033e Plasmodium falciparum 1
23691952 10.1021/np400010c SW480 1
23691952 10.1021/np400010c MCF7 1
23691952 10.1021/np400010c A549 1
23691952 10.1021/np400010c SMMC-7721 1
23691952 10.1021/np400010c HL-60 1

Data from ChEMBL 36 via Core Engine