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Compound Detail

CHEMBL467623

MONURON
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CN(C)C(=O)Nc1ccc(Cl)cc1

Basic Information

ChEMBL ID CHEMBL467623
Name MONURON
Phase Preclinical
Structure Type MOL
InChI Key BMLIZLVNXIYGCK-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

198.7
MW (Da)
2.43
ALogP
1
HBA
1
HBD
32.3
PSA (Ų)
0.74
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C9H11ClN2O
MW 198.65
Aromatic Rings 1
Heavy Atoms 13
NP-Likeness -1.93

Activity Summary

IC50 2 meas. best 6.4

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Photosystem II protein D1
CHEMBL2366481
IC50 6.4 6.4 398.1 1
Photosystem II protein D1
CHEMBL2366463
IC50 5.3 5.3 5011.9 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
- 10.1271/bbb.57.1389 Photosystem II protein D1 2
18834112 10.1021/jm800656v Amine oxidase [flavin-containing] A 1
- 10.1271/bbb.57.1389 No relevant target 1
- 10.1271/bbb.57.1389 Vigna radiata var. radiata 1

Data from ChEMBL 36 via Core Engine