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Compound Detail

CHEMBL474533

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CCN1C(=O)c2c(cc3c(c2O)OCO3)C2=C[C@H](O)[C@@H](O)[C@@H](O)[C@@H]21

Basic Information

ChEMBL ID CHEMBL474533
Phase Preclinical
Structure Type MOL
InChI Key YTQYZKKITXETGV-MBGOOHRESA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
7
Publications
0
Known Names

Molecular Properties

335.3
MW (Da)
-0.56
ALogP
7
HBA
4
HBD
119.7
PSA (Ų)
0.54
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H17NO7
MW 335.31
Aromatic Rings 1
Heavy Atoms 24
NP-Likeness 1.54

Literature References

PubMed DOI Target Context # Activities
19199649 10.1021/jm8013585 PC-3 1
19199649 10.1021/jm8013585 NON-PROTEIN TARGET 1
19199649 10.1021/jm8013585 BXPC-3 1
19199649 10.1021/jm8013585 LoVo 1
19199649 10.1021/jm8013585 A549 1
19199649 10.1021/jm8013585 MCF7 1
19199649 10.1021/jm8013585 No relevant target 1

Data from ChEMBL 36 via Core Engine