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Compound Detail

CHEMBL4795488

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O=C(CCCCC(=O)NC(COCc1cn(CCCc2cn(C[C@@H]3NC[C@@H](O)[C@H]3O)nn2)nn1)(COCc1cn(CCCc2cn(C[C@@H]3NC[C@@H](O)[C@H]3O)nn2)nn1)COCc1cn(CCCc2cn(C[C@@H]3NC[C@@H](O)[C@H]3O)nn2)nn1)NC(COCc1cn(CCCc2cn(C[C@@H]3NC[C@@H](O)[C@H]3O)nn2)nn1)(COCc1cn(CCCc2cn(C[C@@H]3NC[C@@H](O)[C@H]3O)nn2)nn1)COCc1cn(CCCc2cn(C[C@@H]3NC[C@@H](O)[C@H]3O)nn2)nn1

Basic Information

ChEMBL ID CHEMBL4795488
Phase Preclinical
Structure Type MOL
InChI Key HKHNHXVPPORJPS-OTIYRZJJSA-N
0
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

2184.4
MW (Da)

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C92H142N44O20
MW 2184.44

Activity Summary

IC50 2 meas.

Literature References

PubMed DOI Target Context # Activities
32146376 10.1016/j.ejmech.2020.112173 Lysosomal acid glucosylceramidase 1
32146376 10.1016/j.ejmech.2020.112173 Alpha-galactosidase A 1

Data from ChEMBL 36 via Core Engine