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Compound Detail

CHEMBL4848323

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C/C(=N\NC(=O)N1CCC1)c1ccccn1

Basic Information

ChEMBL ID CHEMBL4848323
Phase Preclinical
Structure Type MOL
InChI Key KGHATCWONYIQTN-UKTHLTGXSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

218.3
MW (Da)
1.22
ALogP
3
HBA
1
HBD
57.6
PSA (Ų)
0.60
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C11H14N4O
MW 218.26
Aromatic Rings 1
Heavy Atoms 16
NP-Likeness -2.00

Activity Summary

Kd 1 meas. best 6.36

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
No relevant target
CHEMBL2362975
Kd 6.36 6.36 440.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
No relevant target Kd = 440.0 nM 6.36 Binding affinity to Zn(II)+ incubated for 60 mins using RhodZin-3 by fuorescence... 33538587

Literature References

Data from ChEMBL 36 via Core Engine