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Compound Detail

CHEMBL4850198

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N/C(=N\O)c1cccc(-c2ccc3c(c2)c2cc(-c4cccc(/C(N)=N/O)c4)ccc2n3S(=O)(=O)c2cccc(C(F)(F)F)c2)c1

Basic Information

ChEMBL ID CHEMBL4850198
Phase Preclinical
Structure Type MOL
InChI Key NFPBFUJAIFLGPT-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

643.6
MW (Da)
6.57
ALogP
7
HBA
4
HBD
156.3
PSA (Ų)
0.07
QED
2
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C33H24F3N5O4S
MW 643.65
Aromatic Rings 6
Heavy Atoms 46
NP-Likeness -0.85

Activity Summary

EC50 1 meas. best 5.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
dengue virus type 2
CHEMBL613966
EC50 5.3 5.3 5000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
dengue virus type 2 EC50 = 5000.0 nM 5.3 Antiviral activity against Dengue virus 2 measured at 48 hrs post-infection 34298282

Literature References

PubMed DOI Target Context # Activities
34298282 10.1016/j.ejmech.2021.113695 Genome polyprotein 1
34298282 10.1016/j.ejmech.2021.113695 dengue virus type 2 1

Data from ChEMBL 36 via Core Engine