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Compound Detail

CHEMBL4872708

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CCCCCCNNC(=O)N[C@H]1CC(C(=O)O)=C[C@@H](OC(CC)CC)[C@@H]1NC(C)=O

Basic Information

ChEMBL ID CHEMBL4872708
Phase Preclinical
Structure Type MOL
InChI Key SOEYQILHDYJMSN-IPMKNSEASA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

426.6
MW (Da)
2.23
ALogP
5
HBA
5
HBD
128.8
PSA (Ų)
0.23
QED
0
Ro5 Violations
13
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H38N4O5
MW 426.56
Aromatic Rings 0
Heavy Atoms 30
NP-Likeness 0.48

Activity Summary

IC50 1 meas. best 5.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Neuraminidase
CHEMBL6135
IC50 5.3 5.3 4983.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Neuraminidase IC50 = 4983.0 nM 5.3 Inhibition of Influenza A virus (A/Anhui/1/2005(H5N1) Neuraminidase using MUNANA... 34082224

Literature References

PubMed DOI Target Context # Activities
34082224 10.1016/j.ejmech.2021.113567 Neuraminidase 1

Data from ChEMBL 36 via Core Engine