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Compound Detail

CHEMBL490326

KENGANTHRANOL B
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CC(C)=CCc1c(O)c(CC=C(C)C)c2c(c1O)C(=O)c1c(O)cc(C)c(CC=C(C)C)c1C2O

Basic Information

ChEMBL ID CHEMBL490326
Name KENGANTHRANOL B
Phase Preclinical
Structure Type MOL
InChI Key HAPSTBPDRQRBSO-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

476.6
MW (Da)
6.26
ALogP
5
HBA
4
HBD
98.0
PSA (Ų)
0.37
QED
1
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C30H36O5
MW 476.61
Aromatic Rings 2
Heavy Atoms 35
NP-Likeness 1.58

Activity Summary

IC50 1 meas. best 5.2

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.2 5.2 6300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 6300.0 nM 5.2 Inhibition of Saccharomyces sp. alpha glucosidase by spectrophotometry 16499321

Literature References

PubMed DOI Target Context # Activities
16499321 10.1021/np050407n Unchecked 2

Data from ChEMBL 36 via Core Engine