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Compound Detail

CHEMBL503114

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CC(=O)Nc1nc(C)c(S(=O)(=O)Nc2ccc(C(=O)Nc3ccc4c(c3)N(O)C(=O)/C4=C(\O)c3ccccc3)cc2)s1

Basic Information

ChEMBL ID CHEMBL503114
Phase Preclinical
Structure Type MOL
InChI Key JYXNYOYSNYZAHK-VHXPQNKSSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

605.6
MW (Da)
4.63
ALogP
9
HBA
5
HBD
178.0
PSA (Ų)
0.12
QED
1
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H23N5O7S2
MW 605.65
Aromatic Rings 4
Heavy Atoms 42
NP-Likeness -1.15

Activity Summary

IC50 1 meas. best 4.5

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
unidentified influenza virus
CHEMBL613128
IC50 4.5 4.5 32000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
unidentified influenza virus IC50 = 32000.0 nM 4.5 Antiviral activity against influenza virus 19112024

Literature References

PubMed DOI Target Context # Activities
19112024 10.1016/j.bmc.2008.11.075 unidentified influenza virus 1

Data from ChEMBL 36 via Core Engine