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Compound Detail

CHEMBL50573

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O=C(C1CCCCC1)[C@H]1O[C@H]1[C@@H](O)C1CCCCC1

Basic Information

ChEMBL ID CHEMBL50573
Phase Preclinical
Structure Type MOL
InChI Key QSJPQXTVKNZDHR-CWRNSKLLSA-N
1
Targets
3
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

266.4
MW (Da)
2.84
ALogP
3
HBA
1
HBD
49.8
PSA (Ų)
0.80
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H26O3
MW 266.38
Aromatic Rings 0
Heavy Atoms 19
NP-Likeness 0.52

Activity Summary

IC50 3 meas. best 4.2

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Candida tropicalis
CHEMBL612870
IC50 4.2 4.2 63000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Candida tropicalis IC50 = 63000.0 nM 4.2 Inhibitory activity against Candida tropicalis 16297620

Literature References

PubMed DOI Target Context # Activities
15027875 10.1021/jm0305319 Homo sapiens 1
15027875 10.1021/jm0305319 Plasmodium falciparum 1
16297620 10.1016/j.bmcl.2005.10.101 Candida albicans 1
16297620 10.1016/j.bmcl.2005.10.101 Candida tropicalis 1
16297620 10.1016/j.bmcl.2005.10.101 Pichia kudriavzevii 1

Data from ChEMBL 36 via Core Engine