Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL513383

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
C=CC[C@@H]1C=C[C@H](O/N=C2\[C@H]3CCn4c(=O)n(-c5ccccc5)c(=O)n4[C@H]3[C@H](O)[C@@H]3O[C@H]23)[C@@H](CO)O1

Basic Information

ChEMBL ID CHEMBL513383
Phase Preclinical
Structure Type MOL
InChI Key ZPIPMUZGLPUOCH-NOVIOGFZSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

496.5
MW (Da)
0.14
ALogP
11
HBA
2
HBD
132.7
PSA (Ų)
0.33
QED
1
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H28N4O7
MW 496.52
Aromatic Rings 2
Heavy Atoms 36
NP-Likeness 0.85

Activity Summary

EC50 1 meas. best 5.11

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis C virus
CHEMBL379
EC50 5.11 5.11 7750.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Hepatitis C virus EC50 = 7750.0 nM 5.11 Antiviral activity against HCV replication in human HuH7 cells expressing Rep-Fe... 17682098

Literature References

PubMed DOI Target Context # Activities
17682098 10.1128/aac.00233-07 Hepatitis C virus 1
17682098 10.1128/aac.00233-07 ADMET 1

Data from ChEMBL 36 via Core Engine