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Compound Detail

CHEMBL514105

DICITRININ A
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Cc1c2c(c3oc4cc(=O)c(C)c5c-4c(c3c1O)O[C@H](C)[C@H]5C)O[C@H](C)[C@H]2C

Basic Information

ChEMBL ID CHEMBL514105
Name DICITRININ A
Phase Preclinical
Structure Type MOL
InChI Key WZDGQCYEIYZRBL-NRMKKVEVSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
11
Publications
0
Known Names

Molecular Properties

380.4
MW (Da)
4.99
ALogP
5
HBA
1
HBD
68.9
PSA (Ų)
0.56
QED
0
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C23H24O5
MW 380.44
Aromatic Rings 1
Heavy Atoms 28
NP-Likeness 1.82

Activity Summary

IC50 1 meas. best 4.97

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Radical scavenging activity
CHEMBL613712
IC50 4.97 4.97 10600.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
18281952 10.1021/np0704708 NON-PROTEIN TARGET 1
18281952 10.1021/np0704708 Radical scavenging activity 1
21761866 10.1021/jm200511x HL-60 1
21761866 10.1021/jm200511x HCT-116 1
21761866 10.1021/jm200511x KB 1
26295595 10.1021/acs.jnatprod.5b00450 Aeromonas hydrophila 1
26295595 10.1021/acs.jnatprod.5b00450 Edwardsiella tarda 1
26295595 10.1021/acs.jnatprod.5b00450 Vibrio alginolyticus 1
26295595 10.1021/acs.jnatprod.5b00450 Vibrio anguillarum 1
26295595 10.1021/acs.jnatprod.5b00450 Vibrio harveyi 1
26295595 10.1021/acs.jnatprod.5b00450 Vibrio parahaemolyticus 1

Data from ChEMBL 36 via Core Engine