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Compound Detail

CHEMBL514561

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O=C(/C=C/c1ccccc1Cl)Nc1ccc(C(=O)Nc2ccc3c(c2)N(O)C(=O)/C3=C(\O)c2ccccc2)cc1

Basic Information

ChEMBL ID CHEMBL514561
Phase Preclinical
Structure Type MOL
InChI Key TVPNRHMLBMUNLS-QPKSJOODSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

552.0
MW (Da)
6.41
ALogP
5
HBA
4
HBD
119.0
PSA (Ų)
0.13
QED
2
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C31H22ClN3O5
MW 551.99
Aromatic Rings 4
Heavy Atoms 40
NP-Likeness -0.87

Activity Summary

IC50 1 meas. best 5.02

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
unidentified influenza virus
CHEMBL613128
IC50 5.02 5.02 9500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
unidentified influenza virus IC50 = 9500.0 nM 5.02 Antiviral activity against influenza virus 19112024

Literature References

PubMed DOI Target Context # Activities
19112024 10.1016/j.bmc.2008.11.075 unidentified influenza virus 1

Data from ChEMBL 36 via Core Engine