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Compound Detail

CHEMBL517863

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COc1cc([C@H]2OC[C@]3(O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)[C@@H](c4ccc(O)c(OC)c4)OC[C@H]23)ccc1O

Basic Information

ChEMBL ID CHEMBL517863
Phase Preclinical
Structure Type MOL
InChI Key DRAPQDCEBKBPQE-ACFZRETJSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

536.5
MW (Da)
0.13
ALogP
12
HBA
6
HBD
176.8
PSA (Ų)
0.28
QED
3
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C26H32O12
MW 536.53
Aromatic Rings 2
Heavy Atoms 38
NP-Likeness 1.86

Activity Summary

IC50 1 meas. best 4.69

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Radical scavenging activity
CHEMBL613712
IC50 4.69 4.69 20300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
11473417 10.1021/np0100845 NON-PROTEIN TARGET 3
11473417 10.1021/np0100845 Radical scavenging activity 1

Data from ChEMBL 36 via Core Engine