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Compound Detail

CHEMBL5395744

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C=CC(=O)Nc1cccc(Nc2nc(N3CCCC[C@H]3CCO)nc3c2ncn3CC)c1

Basic Information

ChEMBL ID CHEMBL5395744
Phase Preclinical
Structure Type MOL
InChI Key NDYGLDMFZGWJMX-SFHVURJKSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

435.5
MW (Da)
3.46
ALogP
8
HBA
3
HBD
108.2
PSA (Ų)
0.47
QED
0
Ro5 Violations
8
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C23H29N7O2
MW 435.53
Aromatic Rings 3
Heavy Atoms 32
NP-Likeness -1.01

Activity Summary

IC50 2 meas. best 8.1

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 8.1 8.1 8.0 1
Lung cancer cell line
CHEMBL614790
IC50 8.1 8.1 8.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
37731700 10.1039/d3md00004d Unchecked 1
37731700 10.1039/d3md00004d Lung cancer cell line 1

Data from ChEMBL 36 via Core Engine