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Compound Detail

CHEMBL5401545

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CCC(CC)O[C@@H]1C=C(P(=O)(O)O[C@H]2[C@@H](O)[C@@H](CO)O[C@@H](OC)[C@@H]2O)C[C@H](N)[C@H]1NC(C)=O

Basic Information

ChEMBL ID CHEMBL5401545
Phase Preclinical
Structure Type MOL
InChI Key SASAWRLEIBZULD-NOVIIDPASA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

496.5
MW (Da)
-0.66
ALogP
10
HBA
6
HBD
190.0
PSA (Ų)
0.21
QED
1
Ro5 Violations
10
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H37N2O10P
MW 496.49
Aromatic Rings 0
Heavy Atoms 33
NP-Likeness 1.66

Activity Summary

Ki 1 meas. best 9.54

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Neuraminidase
CHEMBL2051
Ki 9.54 9.54 0.3 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Neuraminidase Ki = 0.29 nM 9.54 Binding affinity to influenza A virus H1N1 (A/Norway/1758/07) neuraminidase usin... 37120995

Literature References

PubMed DOI Target Context # Activities
37120995 10.1016/j.ejmech.2023.115410 Neuraminidase 1

Data from ChEMBL 36 via Core Engine