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Compound Detail

CHEMBL5411309

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CC(=O)N[C@H]1[C@H]([C@H](O)[C@H](O)CO)O[C@H](S(=O)(=O)O)C[C@@H]1O

Basic Information

ChEMBL ID CHEMBL5411309
Phase Preclinical
Structure Type MOL
InChI Key VZXYJUJTPRTNBD-IHICSVBISA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

329.3
MW (Da)
-3.43
ALogP
8
HBA
6
HBD
173.6
PSA (Ų)
0.28
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H19NO9S
MW 329.33
Aromatic Rings 0
Heavy Atoms 21
NP-Likeness 1.06

Activity Summary

IC50 1 meas. best 5.05

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Neuraminidase
CHEMBL3232678
IC50 5.05 5.05 8860.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Neuraminidase IC50 = 8860.0 nM 5.05 Inhibition of influenza A virus A/RI/5+/1957(H2N2) neuraminidase using 4-MU-Neu5... 37120995

Literature References

PubMed DOI Target Context # Activities
37120995 10.1016/j.ejmech.2023.115410 Neuraminidase 1

Data from ChEMBL 36 via Core Engine