Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL5417969

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
Cc1[nH]c(C(=O)Nc2nc3c(OC(C[N+](C)(C)C)c4ccccc4)cc(C(=O)O)cc3s2)c(Cl)c1Cl.[I-]

Basic Information

ChEMBL ID CHEMBL5417969
Phase Preclinical
Structure Type MOL
InChI Key RTDXFXCNZDOECC-UHFFFAOYSA-N
Parent Compound CHEMBL5499458
Active Moiety CHEMBL5499458
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
8
Publications
0
Known Names

Molecular Properties

548.5
MW (Da)
6.02
ALogP
5
HBA
3
HBD
104.3
PSA (Ų)
0.23
QED
2
Ro5 Violations
8
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H25Cl2IN4O4S
MW 675.38
Aromatic Rings 4
Heavy Atoms 36
NP-Likeness -0.94

Literature References

PubMed DOI Target Context # Activities
36634346 10.1021/acs.jmedchem.2c01597 Unchecked 5
36634346 10.1021/acs.jmedchem.2c01597 Escherichia coli 2
36634346 10.1021/acs.jmedchem.2c01597 Acinetobacter baumannii 2
36634346 10.1021/acs.jmedchem.2c01597 Pseudomonas aeruginosa 2
36634346 10.1021/acs.jmedchem.2c01597 Staphylococcus aureus 1
36634346 10.1021/acs.jmedchem.2c01597 DNA gyrase subunit B 1
36634346 10.1021/acs.jmedchem.2c01597 No relevant target 1
36634346 10.1021/acs.jmedchem.2c01597 ADMET 1

Data from ChEMBL 36 via Core Engine