Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL5571121

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
O=C(Cc1ccccc1Nc1c(Cl)cccc1Cl)N/N=C1\C(=O)N(Cc2ccccc2)c2ccccc21

Basic Information

ChEMBL ID CHEMBL5571121
Phase Preclinical
Structure Type MOL
InChI Key MILFNWMXOQXGFV-YLHCSOALSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

529.4
MW (Da)
6.35
ALogP
4
HBA
2
HBD
73.8
PSA (Ų)
0.27
QED
2
Ro5 Violations
7
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C29H22Cl2N4O2
MW 529.43
Aromatic Rings 4
Heavy Atoms 37
NP-Likeness -1.42

Activity Summary

IC50 1 meas. best 5.18

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.18 5.18 6640.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 6640.0 nM 5.18 Inhibition of soybean 15-LOX 37862815

Literature References

PubMed DOI Target Context # Activities
37862815 10.1016/j.ejmech.2023.115866 Unchecked 1

Data from ChEMBL 36 via Core Engine