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Compound Detail

CHEMBL5591152

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C=C1C(=O)O[C@H]2[C@H]1C(COC(=O)CC(C)(C)CC(=O)O)C/C=C\CC[C@@]1(C)O[C@@H]21

Basic Information

ChEMBL ID CHEMBL5591152
Phase Preclinical
Structure Type MOL
InChI Key YBILUBZCZRFXEU-KXDGSLRASA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

406.5
MW (Da)
3.03
ALogP
6
HBA
1
HBD
102.4
PSA (Ų)
0.31
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H30O7
MW 406.48
Aromatic Rings 0
Heavy Atoms 29
NP-Likeness 2.35

Activity Summary

IC50 1 meas. best 4.44

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
MDA-MB-231
CHEMBL400
IC50 4.44 4.44 36400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
MDA-MB-231 IC50 = 36400.0 nM 4.44 Antiproliferative activity against human MDA-MB-231 cells assessed as inhibition... 38104376

Literature References

PubMed DOI Target Context # Activities
38104376 10.1016/j.ejmech.2023.116024 MDA-MB-231 1

Data from ChEMBL 36 via Core Engine