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Compound Detail

CHEMBL5595207

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O=C(Cc1ccccc1Nc1c(Cl)cccc1Cl)N/N=C1\C(=O)N(Cc2ccccc2)c2ccc(Cl)cc21

Basic Information

ChEMBL ID CHEMBL5595207
Phase Preclinical
Structure Type MOL
InChI Key VAVCLYIUGPQYRL-LSWMGQQCSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

563.9
MW (Da)
7.00
ALogP
4
HBA
2
HBD
73.8
PSA (Ų)
0.24
QED
2
Ro5 Violations
7
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C29H21Cl3N4O2
MW 563.87
Aromatic Rings 4
Heavy Atoms 38
NP-Likeness -1.50

Activity Summary

IC50 1 meas. best 5.34

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.34 5.34 4610.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 4610.0 nM 5.34 Inhibition of soybean 15-LOX 37862815

Literature References

PubMed DOI Target Context # Activities
37862815 10.1016/j.ejmech.2023.115866 Unchecked 1

Data from ChEMBL 36 via Core Engine