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Compound Detail

CHEMBL5595575

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N#CCNC(=O)c1ccc(-c2ccnc(Nc3ccc(N4CCC(C(=O)NCCCCCC#Cc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)n2)cc1

Basic Information

ChEMBL ID CHEMBL5595575
Phase Preclinical
Structure Type MOL
InChI Key ZFFKARYWSKLSMW-UHFFFAOYSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

805.9
MW (Da)
4.49
ALogP
11
HBA
4
HBD
206.6
PSA (Ų)
0.06
QED
2
Ro5 Violations
13
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C45H43N9O6
MW 805.90
Aromatic Rings 4
Heavy Atoms 60
NP-Likeness -1.09

Literature References

PubMed DOI Target Context # Activities
38838918 10.1016/j.bmcl.2024.129838 HEL 1
38838918 10.1016/j.bmcl.2024.129838 K562 1
38838918 10.1016/j.bmcl.2024.129838 Tyrosine-protein kinase JAK1 1
38838918 10.1016/j.bmcl.2024.129838 Protein cereblon/JAK1 1
38838918 10.1016/j.bmcl.2024.129838 Protein cereblon/Tyrosine-protein kinase JAK2 1
38838918 10.1016/j.bmcl.2024.129838 THP-1 1

Data from ChEMBL 36 via Core Engine