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Compound Detail

CHEMBL5745979

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CC12CCC3c4ccc(O)cc4CC(CCCCCCCCC[S+]([O-])CCCC(F)(F)C(F)(F)F)C3C1CCC2O

Basic Information

ChEMBL ID CHEMBL5745979
Phase Preclinical
Structure Type MOL
InChI Key VWUXBMIQPBEWFH-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

606.8
MW (Da)
8.68
ALogP
3
HBA
2
HBD
63.5
PSA (Ų)
0.13
QED
2
Ro5 Violations
14
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C32H47F5O3S
MW 606.78
Aromatic Rings 1
Heavy Atoms 41
NP-Likeness 1.48

Activity Summary

IC50 1 meas. best 8.64

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 8.64 8.64 2.3 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 2.29 nM 8.64 LanthaScreen Competitive Binding Assay: Compounds were screened for their abilit... -

Data from ChEMBL 36 via Core Engine