Compound Detail
CHEMBL5784483
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Basic Information
| ChEMBL ID | CHEMBL5784483 |
| Phase | Preclinical |
| Structure Type | MOL |
| InChI Key | QJTKHFUSFJUINE-IBGZPJMESA-N |
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names
Molecular Properties
367.2
MW (Da)
Drug Information
| Availability | Unknown |
| Chirality | Unknown |
Activity Summary
IC50 1 meas. best 6.56
Target Activity Profile
| Target | Type | Best pChEMBL | Mean pChEMBL | Best (nM) | # Data |
|---|---|---|---|---|---|
| Proteasome Macropain subunit MB1 CHEMBL4662 | IC50 | 6.56 | 6.56 | 275.0 | 1 |
Activity Data Samples
Top measurements by pChEMBL value
| Target | Type | Rel. | Value | Units | pChEMBL | Assay | PubMed |
|---|---|---|---|---|---|---|---|
| Proteasome Macropain subunit MB1 | IC50 | = | 275.0 | nM | 6.56 | Determination of Beta5 Activity: Measurement of Beta5 inhibition is performed in... | - |
Data from ChEMBL 36 via Core Engine