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Compound Detail

CHEMBL5917491

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NS(=O)(=O)OC[C@H]1C[C@@H](Nc2ccnc3cc(-c4cccc(-c5ccccc5)c4)nn23)[C@H](O)[C@@H]1O

Basic Information

ChEMBL ID CHEMBL5917491
Phase Preclinical
Structure Type MOL
InChI Key OHUBWOCZKZLWIV-ILEGPTGMSA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

495.6
MW (Da)
1.81
ALogP
9
HBA
4
HBD
152.1
PSA (Ų)
0.30
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C24H25N5O5S
MW 495.56
Aromatic Rings 4
Heavy Atoms 35
NP-Likeness -0.50

Data from ChEMBL 36 via Core Engine