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Compound Detail

CHEMBL5933555

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COc1ccc2nn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@@H]6[C@H]5CC[C@]34C)nc2c1

Basic Information

ChEMBL ID CHEMBL5933555
Phase Preclinical
Structure Type MOL
InChI Key SZQDGVNMPGIAJV-CCZABAJOSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

465.6
MW (Da)
5.03
ALogP
6
HBA
1
HBD
77.2
PSA (Ų)
0.69
QED
1
Ro5 Violations
4
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H39N3O3
MW 465.64
Aromatic Rings 2
Heavy Atoms 34
NP-Likeness 0.85

Activity Summary

IC50 1 meas. best 7.52

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 7.52 7.52 30.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 30.0 nM 7.52 Steroid Inhibition of TBPS Binding: TBPS binding assays using rat brain cortical... -

Data from ChEMBL 36 via Core Engine