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Compound Detail

CHEMBL5938995

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Cn1c(CSc2nonc2/C(=N/O)Nc2ccc(F)c(Br)c2)n[nH]c1=O

Basic Information

ChEMBL ID CHEMBL5938995
Phase Preclinical
Structure Type MOL
InChI Key HMWGCTYZYICOLX-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

444.2
MW (Da)
1.93
ALogP
9
HBA
3
HBD
134.2
PSA (Ų)
0.18
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H11BrFN7O3S
MW 444.25
Aromatic Rings 3
Heavy Atoms 26
NP-Likeness -2.17

Activity Summary

IC50 1 meas. best 7.42

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Indoleamine 2,3-dioxygenase 1
CHEMBL4685
IC50 7.42 7.42 37.8 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Indoleamine 2,3-dioxygenase 1 IC50 = 37.8 nM 7.42 Enzyme Assay: HIS-tagged IDO1 protein was recombinantly expressed in Escherichia... -

Data from ChEMBL 36 via Core Engine