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Compound Detail

CHEMBL5964175

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C[C@@]1(O)CC[C@H]2[C@H](CC[C@@H]3[C@@H]2CC[C@]2(C)[C@@H](C(=O)Cc4nccc5ccccc45)CC[C@@H]32)C1

Basic Information

ChEMBL ID CHEMBL5964175
Phase Preclinical
Structure Type MOL
InChI Key VAFZCEGZEXWGBW-WRAPKJGWSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

445.6
MW (Da)
6.37
ALogP
3
HBA
1
HBD
50.2
PSA (Ų)
0.60
QED
1
Ro5 Violations
3
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C30H39NO2
MW 445.65
Aromatic Rings 2
Heavy Atoms 33
NP-Likeness 1.24

Activity Summary

IC50 1 meas. best 6.52

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.52 6.52 300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 300.0 nM 6.52 Steroid Inhibition of TBPS Binding: TBPS binding assays using rat brain cortical... -

Data from ChEMBL 36 via Core Engine