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Compound Detail

CHEMBL5973780

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Cc1ccc(-c2ccc(-c3cccc(-c4nn(-c5nc(C(=O)O)cs5)c(CC5CC5)c4Cc4ccc(S(N)(=O)=O)c(F)c4)c3)cc2)s1

Basic Information

ChEMBL ID CHEMBL5973780
Phase Preclinical
Structure Type MOL
InChI Key OQDIDGGIMKHMBH-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

684.8
MW (Da)
7.73
ALogP
8
HBA
2
HBD
128.2
PSA (Ų)
0.15
QED
2
Ro5 Violations
10
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C35H29FN4O4S3
MW 684.84
Aromatic Rings 6
Heavy Atoms 47
NP-Likeness -1.37

Activity Summary

IC50 1 meas. best 6.26

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.26 6.26 550.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 550.0 nM 6.26 Biochemical Assay: Test compounds were placed in a Greiner Bio-One (Monroe, N.C.... -

Data from ChEMBL 36 via Core Engine