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Compound Detail

CHEMBL6024856

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C[C@]12CC[C@H]3[C@@H](CC[C@H]4C[C@@](O)(CF)CC[C@@H]43)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2ccccc21

Basic Information

ChEMBL ID CHEMBL6024856
Phase Preclinical
Structure Type MOL
InChI Key SRNDDAGADSAVAP-AECCJQPVSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

453.6
MW (Da)
4.97
ALogP
5
HBA
1
HBD
68.0
PSA (Ų)
0.71
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C27H36FN3O2
MW 453.60
Aromatic Rings 2
Heavy Atoms 33
NP-Likeness 0.42

Activity Summary

IC50 1 meas. best 6.52

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.52 6.52 300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 300.0 nM 6.52 Steroid Inhibition of TBPS Binding: TBPS binding assays using rat brain cortical... -

Data from ChEMBL 36 via Core Engine