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Compound Detail

CHEMBL6033400

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COc1cc(C(=O)Nc2nnc(-c3ccncc3)s2)ccc1OCc1ccc(F)cc1

Basic Information

ChEMBL ID CHEMBL6033400
Phase Preclinical
Structure Type MOL
InChI Key KEWVGNGIYAOJRP-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

436.5
MW (Da)
4.58
ALogP
7
HBA
1
HBD
86.2
PSA (Ų)
0.46
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H17FN4O3S
MW 436.47
Aromatic Rings 4
Heavy Atoms 31
NP-Likeness -1.78

Activity Summary

Ki 1 meas. best 7.85

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NADPH oxidase 1
CHEMBL1287628
Ki 7.85 7.85 14.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NADPH oxidase 1 Ki = 14.0 nM 7.85 ROS Production Measurement on hNOX1 Membranes: All solutions were placed on ice ... -

Data from ChEMBL 36 via Core Engine