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Compound Detail

CHEMBL6068328

ELTROMBOPAG CHOLINE
💊 Approved Drug
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💊 Approved Drug
CC1=NN(c2ccc(C)c(C)c2)C(=O)/C1=N\Nc1cccc(-c2cccc(C(=O)[O-])c2)c1O.C[N+](C)(C)CCO

Basic Information

ChEMBL ID CHEMBL6068328
Name ELTROMBOPAG CHOLINE
Phase Approved
Structure Type MOL
InChI Key XSHFVAAXJHNDKZ-OUFJFOJPSA-M
Therapeutic ✓ Yes
Parent Compound CHEMBL461101
Active Moiety CHEMBL461101

Known Names

Alvaiz Eltrombopag choline
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
0
Publications
2
Known Names
4
Indications
1
Mechanisms

Molecular Properties

442.5
MW (Da)
4.56
ALogP
6
HBA
3
HBD
114.6
PSA (Ų)
0.40
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
First Approval 2023
Availability Prescription
Chirality Achiral

Routes of Administration

Oral

Flags

Black Box Warning
USAN Stem -trombopag

Extended Properties

Molecular Formula C30H35N5O5
MW 545.64
Aromatic Rings 3
Heavy Atoms 33
NP-Likeness -1.07

Mechanism of Action

Mechanism Action Type Target Direct Efficacy
Thrombopoietin receptor agonist AGONIST Thrombopoietin receptor

Indications

Anemia, Aplastic Hepatitis C, Chronic Purpura, Thrombocytopenic, Idiopathic Thrombocytopenia

Drug Warnings

Black Box Warning
General Warning
Country: United States

Data from ChEMBL 36 via Core Engine