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Compound Detail

CHEMBL6070359

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C[C@@](O/N=C(\C(=O)N[C@@H]1C(=O)N2C(C(=O)O)=C(CSCCNC(=O)c3ccc(O)c(O)c3Cl)CS[C@H]12)c1nc(N)sc1Cl)(C(=O)O)C(F)(F)F

Basic Information

ChEMBL ID CHEMBL6070359
Phase Preclinical
Structure Type MOL
InChI Key CYULNAKMYJBZIR-YPZWEWQISA-N
0
Targets
0
Activities
0
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

803.6
MW (Da)
2.47
ALogP
14
HBA
7
HBD
254.1
PSA (Ų)
0.05
QED
3
Ro5 Violations
13
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C26H23Cl2F3N6O10S3
MW 803.60
Aromatic Rings 2
Heavy Atoms 50
NP-Likeness -0.38

Data from ChEMBL 36 via Core Engine