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Compound Detail

CHEMBL68672

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CCN(CC)C(=O)/C=C/c1ccc(O)c(O)c1

Basic Information

ChEMBL ID CHEMBL68672
Phase Preclinical
Structure Type MOL
InChI Key IVRFYKXAGRJRNP-SOFGYWHQSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
9
Publications
0
Known Names

Molecular Properties

235.3
MW (Da)
1.98
ALogP
3
HBA
2
HBD
60.8
PSA (Ų)
0.62
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H17NO3
MW 235.28
Aromatic Rings 1
Heavy Atoms 17
NP-Likeness 0.07

Activity Summary

IC50 2 meas. best 5.39

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.39 5.39 4100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 4100.0 nM 5.39 Evaluated for the antioxidant property by measuring the inhibition of microsomal... 11206462

Literature References

PubMed DOI Target Context # Activities
34157569 10.1016/j.bmc.2021.116247 Amyloid-beta precursor protein 3
11206462 10.1016/s0960-894x(00)00630-2 Unchecked 1
17596944 10.1016/j.bmcl.2007.06.016 Tyrosine-protein phosphatase non-receptor type 1 1
20181415 10.1016/j.ejmech.2010.01.066 Bacillus subtilis 1
20181415 10.1016/j.ejmech.2010.01.066 Pseudomonas fluorescens 1
20181415 10.1016/j.ejmech.2010.01.066 Staphylococcus aureus 1
20181415 10.1016/j.ejmech.2010.01.066 Candida albicans 1
30347330 10.1016/j.ejmech.2018.10.025 Tyrosinase 1
30347330 10.1016/j.ejmech.2018.10.025 No relevant target 1

Data from ChEMBL 36 via Core Engine