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Compound Detail

CHEMBL72695

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CCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(=O)O)NC(C)=O)[C@@H](C)CC)C(C)C)C(=O)O

Basic Information

ChEMBL ID CHEMBL72695
Phase Preclinical
Structure Type BOTH
InChI Key NELACTXYCHECFZ-DZQZDKHXSA-N
0
Targets
5
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

698.8
MW (Da)
-1.04
ALogP
9
HBA
8
HBD
277.7
PSA (Ų)
0.08
QED
2
Ro5 Violations
20
Rot. Bonds

Drug Information

Molecule Type Protein
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C31H50N6O12
MW 698.77
Aromatic Rings 0
Heavy Atoms 49
NP-Likeness -0.01

Activity Summary

IC50 5 meas.

Literature References

PubMed DOI Target Context # Activities
15239657 10.1021/jm049864b NS3 1
9873610 10.1016/s0960-894x(98)00480-6 Hepatitis C virus serine protease, NS3/NS4A 1
11055335 10.1016/s0960-894x(00)00465-0 NS3 1
14695826 10.1021/jm0303002 Unchecked 1
27501244 10.1021/acs.jmedchem.6b00915 Hepatitis C virus serine protease, NS3/NS4A 1

Data from ChEMBL 36 via Core Engine